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Abstract LB242: Discovery and characterization of BRSD-143, an orally bioavailable panKRAS inhibitor

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Year: 2025
Type: conference-abstract
Source: Cancer Research
DOI: 10.1158/1538-7445.am2025-lb242
Authors: Charles Y. Cho, Qian Liu, Jun Liu, Deborah A. Knee, David P. Kodack, Dean P. Phillips, Phillip B. Alper, Hong Jin, Wendy Richmond, Sarah E. Kochanek, Hong Yin, Yu Chen, Jie Li, Cyrus Virata, David H. Jones, Jose C. Juarez, Michael DiDonato, Brandon L. Taylor, Dmitry Borkin, Dong Han, Xianzhong Liu, Vicki W. Zhou, Lilin Li, Rita Das, Varunika Vivekanandan, Flavio Somanji, David A. Ruddy, Michelle Piquet, Miriam Coor, Eiru Kim, Yelena Sarkisova, Min Lu, Guoxun Liu, Danielle Roman, William P. Gordon, Todd Groessl, Michael Shapiro, Yvonne Wang, Darbi Witmer, Agnes Vidal-Biggart, Yong Jia, Jacob R. Haling
Institution: Novartis (Switzerland)
Language: English

Topic: Protein Kinase Regulation and GTPase Signaling
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W4409820763
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Related to: 10
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