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Residue-Selective Inhibitors Discovery via Covalent DNA-Encoded Chemical Libraries with Diverse Warheads

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Year: 2025
Type: article
Source: Journal of the American Chemical Society
DOI: 10.1021/jacs.5c01712
Authors: Xinyuan Wu, Jiayi Pan, Rufeng Fan, Yiwei Zhang, Chao Wang, Guoliang Wang, Jiaxiang Liu, Mengqing Cui, Jinfeng Yue, Rui Jin, Zhiqiang Duan, Mingyue Zheng, Lianghe Mei, Lu Zhou, Minjia Tan, Jing Ai, Xiaojie Lu
Institutions: Chinese Academy of Sciences, Shanghai Institute of Materia Medica, University of Chinese Academy of Sciences, State Key Laboratory of Drug Research, Nanjing University of Chinese Medicine, Fudan University
Language: English

Topic: Chemical Synthesis and Analysis
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences

Open Access status: closed

Funders: Innovative Research Team of High-level Local University in Shanghai, National Natural Science Foundation of China, Chinese Academy of Sciences, Shanghai Institute of Materia Medica, Chinese Academy of Sciences
Awards: G113098703, G3215655507, G333480629, G3999105043, G4778903190, G607916541, G6390070855, G6592492841, G8012778378
OpenAlex ID: W4409869802
FWCI: 8.616
Cites: 67
Cited by: 33
Related to: 10
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