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Lysine‐Targeting, Covalent Inhibitors of Bromodomain BD1 of BET Proteins in Live Cells and Animals

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Year: 2025
Type: article
Source: Angewandte Chemie
DOI: 10.1002/ange.202424832
Authors: Tao Li, Wenjie Zhang, Yiqing Wang, Guangyu Xu, Fengfei Miao, Peng Chen, Guanghui Tang, Xiaotong Ze, Jing Xiang, Jiaqian Yan, Miaomiao Wang, Min Liu, Xiaojie Wang, Wei Tang, Fan Yi, Zhi‐Min Zhang, Rui Wang, Shao Q Yao, Yusheng Xie
Institutions: Shandong University, Jinan University, National University of Singapore, Second Hospital of Shandong University, Shenzhen Bay Laboratory
Language: English

Topic: Protein Degradation and Inhibitors
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: National Natural Science Foundation of China, National Medical Research Council, Shenzhen Science and Technology Innovation Program
Awards: G4229283544, G8194676655, G8614504637, G9188717
OpenAlex ID: W4410039875
FWCI: 0.261
Cites: 60
Cited by: 1
Related to: 10
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