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Discovery of Tamsulosin Derivatives with Shifted Selectivity from the α1-Adrenergic Receptor to ANO1 as Potent Antiosteoporotic Agents

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Year: 2025
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.5c01408
Authors: Chaoquan Tian, Weijia Sun, Tao Yu, Shuai Guo, Yiqing Zhang, Shuang Li, Shuang Li, Jiaqi He, Mingqi Yu, Lingkang Wu, Wenyi Mei, Yuheng Li, Yuheng Li, Zhenjiang Zhao, Lili Zhu, Yanyan Diao, Honglin Li, Yingxian Li, Yingxian Li, Shiliang Li, Shiliang Li
Institutions: East China University of Science and Technology, Beijing Institute of Technology, China Astronaut Research and Training Center, East China Normal University, Hebei University, Fudan University, Huadong Hospital
Language: English

Topic: Bone Metabolism and Diseases
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: National Natural Science Foundation of China, China Postdoctoral Science Foundation, Shanghai Rising-Star Program, National Key Research and Development Program of China
Awards: G1404193024, G1440936925, G1618279006, G2181064121, G5009833721, G5038972950, G5636376179, G8796382498
OpenAlex ID: W4413103659
FWCI:
Cites: 33
Cited by:
Related to: 10
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