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Selectivity Profiling of Bromodomain PROTACs Using Chemical Inducers of Proximity DNA-Encoded Library Screening

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Year: 2025
Type: article
Source: ACS Chemical Biology
DOI: 10.1021/acschembio.5c00413
Authors: Yuen Ting Chow, Bingqi Tong, Zher Yin Tan, Antonin Tutter, Zhihan Nan, Patricia A. Horton, Michael J. Romanowski, Frédéric J. Zécri, Stuart L. Schreiber, Shuang Liu
Institutions: Broad Institute, Harvard University
Language: English

Topic: Protein Degradation and Inhibitors
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences

Open Access status: closed

Funders: Agency for Science, Technology and Research, National Cancer Institute, National Institute of General Medical Sciences
Awards: G3844817483, G5102869059, G6041155856
OpenAlex ID: W4413108046
FWCI: 1.305
Cites: 28
Cited by: 5
Related to: 10
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