In Pursuit of Best-in-Class MCL-1 Inhibitors: Discovery of Highly Potent 1,4-Indoyl Macrocycles with Favorable Physicochemical Properties
Year: 2025
Type: article
Source: Journal of Medicinal Chemistry
Authors: Ingrid Adriana Velter, William Lento, Aldo Peschiulli, Tristan D. Reuillon, Sofia Ferrer, Sergio Orgaz-Gordillo, Peter Buijnsters, Benoît C. A. G. De Boeck, Samuel Demin, Yves Van Roosbroeck, Matthieu Jouffroy, Ann Vos, Bradley Miller, Paul Shaffer, Seong Joo Koo, Maria Dominguez Blanco, Lisa McQueen, Cristina Altrocchi, Ruud Bueters, Petra Vinken, Mariette Bekkers, Helena Steyvers, Christina Guttke, David Walker, Marcus Bauser, David M. Wilson, Ulrike Philippar, Frederik J. R. Rombouts
Language: English
Subfield: Molecular Biology
Domain: Life Sciences
Open Access status: closed
OpenAlex ID: W4413276519
