Development of Scalable Synthesis of Chiral Sultam via a Chiral Phosphoric Acid-Promoted tert-Butyl Carbamate Deprotection–Resolution Sequence or Diastereoselective Hydrogenation
Year: 2025
Type: article
Authors: Caroline A. Blakemore, Adam R. Brown, Todd W. Butler, Christopher W. am Ende, Nahian Khan, Sarai Lara-Boykin, Bryan Li, Guochun Ma, Javier Magano, Subham Mahapatra, Peter D. Morse, Giselle P. Reyes, Colin Rose, Neal W. Sach, Liam S. Sharninghausen, Jared Van Haitsma, Pengzhi Wang, Daniel W. Widlicka, Zebediah C. Girvin
Institutions: Pfizer (United States), Pharmaron (China)
Language: English
Subfield: Organic Chemistry
Field: Chemistry
Domain: Physical Sciences
Open Access status: closed
OpenAlex ID: W4414163151
