Dual-regioselective direct C(sp 2 )-arylation of unprotected β-enamino esters with 2-indolylmethanols catalyzed by Brønsted acid
Year: 2025
Type: article
Abstract: An dual-regioselective strategy has been developed for the direct C(sp 2 )-arylation of β -enamino esters with 2-indolylmethanols, delivering 48 structurally diverse indole-enamino ester hybrids in moderate to excellent yields (up to 98%).
Source: RSC Advances
DOI: 10.1039/d5ra05581d
Authors: Qing-Chun Song, Pei-Hua Zhao, Yu-Xi Xing, Chen-Xin Bao, Ling-Yan Chen, Ya Li
Institutions: Shanghai University of Engineering Science, Xiamen University
Language: English
Subfield: Organic Chemistry
Field: Chemistry
Domain: Physical Sciences
Open Access status: gold
Estimated APC paid: $1,042
OpenAlex ID: W4414661077