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Lipophilicity-Optimized PARP-1 Tracers: Minimizing Hepatic Retention for Enhanced Target-to-Background PET Imaging

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Year: 2025
Type: article
Source: Molecular Pharmaceutics
DOI: 10.1021/acs.molpharmaceut.5c01089
Authors: Yi Xie, Chongchong Gao, Hualong Chen, Xuebo Cheng, Xinyu Sun, Yajing Liu, Futao Liu, Zehui Wu
Institutions: Army Medical University, Capital Medical University, Daping Hospital, Beijing Institute for Brain Disorders, National Medical Products Administration, Peking University Cancer Hospital
Language: English

Topic: Radiopharmaceutical Chemistry and Applications
Subfield: Radiology, Nuclear Medicine and Imaging
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: National Natural Science Foundation of China, Beijing Municipal Natural Science Foundation
Awards: G1255891816, G2509203876, G4732197427, G6320720502
OpenAlex ID: W4414948113
FWCI: 3.197
Cites: 28
Cited by: 6
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