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Structural Optimization of Bicyclic Oxo-Boronates as Dual Metallo- and Serine-β-Lactamase Inhibitors

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Year: 2025
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.5c02230
Authors: Zeng-Bao Yang, Si-Qi Wei, Yao-Geng Wang, Xiang-Min Dong, Hao-Xiang Xu, Xiao-Lan Li, Jian Peng, Rui-Chuan Yin, Guo-Bo Li
Institution: Sichuan University
Language: English

Topic: Antibiotic Resistance in Bacteria
Subfield: Molecular Medicine
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: National Natural Science Foundation of China, Natural Science Foundation of Sichuan Province, Sichuan Province Science and Technology Support Program, National Key Research and Development Program of China
Awards: G2432285787, G3441359491, G6446954825, G658642563, G683695221, G7301097705, G7771303265, G8434933821
OpenAlex ID: W4415109060
FWCI: 0.955
Cites: 51
Cited by: 4
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