Design, Synthesis, and T Cell Checkpoint Combination Potential Of First-In-Class DGKα/ζ Inhibitor BMS-986408
Year: 2025
Type: article
Source: Journal of Medicinal Chemistry
Authors: Denise C. Grünenfelder, Upender Velaparthi, Jayakumar S. Warrier, Louis Chupak, Chetan Padmakar Darne, Bireshwar Dasgupta, T. G. Murali Dhar, Min Ding, Robert Gentles, Yazhong Huang, Prasada R. Jalagam, Manjunatha Narayana Rao Kamble, Raju Mannoori, Scott Martin, Shana L. Posy, Hasibur Rahaman, Thiruvenkadam Raja, Kotha Rathnakar Reddy, Saumya Roy, Amy Sarjeant, John S. Tokarski, Gopikishan Tonukunuru, Sivasudar Velaiah, Xiaofan Zheng, Aravind Anandam, Gopal Dhar, Shailesh Dudhgaonkar, R. Marcus Fancher, Siddheshwar Layane, Si-Qi Liu, Swagatam Ray, Hongchen Qiu, Susan Wee, Sagnik Chatterjee, Myrtle Davis, Elizabeth Dierks, Anoop Kumar, Thanga Mariappan, Robin Moore, Bokka Venkata Murali, Ramola Sane, Dana Banas, Deepa Calambur, Erica Cook, Priya Dehal, Hua Fang, Gregory Locke, Joseph G. Naglich, Madhu Sudhan Ravindran, Lumelle Schneeweis, Debarati M. Tagore, Mark Witmer, Abigail E. Witt, Dianlin Xie, Emma Lees, Michael Wichroski, Nicholas A. Meanwell, Robert Borzilleri, Richard E. Olson
Language: English
Subfield: Oncology
Field: Medicine
Domain: Health Sciences
Open Access status: closed
OpenAlex ID: W4415148597
