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Discovery of NP3-742: A Structurally Diverse NLRP3 Inhibitor Identified through an Unusual Phenol Replacement

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Year: 2025
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.5c02412
Authors: Juraj Velcicky, Jean-Baptiste Langlois, Michael Wright, Philipp Janser, Daniela Angst, Christelle Arnold, Karen Beltz, Silke Brenneisen, Celine Dubois, Janet Dawson, Christian Fischer, Nina Gommermann, Andreas Heizmann, Slavica Ilic, Rainer Machauer, Magdalena Maschlej, Sarah Monnerat, Daniel Pflieger, Jacinda Ristov, Joelle Rubert, Günther Schwalm, Daniel R. Smith, Honnappa Srinivas, Roland Steiner, Aleksandar Stojanovic, Thomas Troxler, Adeline Unterreiner, Eric Vangrevelinghe, Nicole von Burg, Jennifer Wunderlich, Christopher J. Farady, Angela Mackay
Institutions: Novartis (Switzerland), Novartis Institutes for BioMedical Research
Language: English

Topic: Inflammasome and immune disorders
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W4415224941
FWCI: 2.089
Cites: 67
Cited by: 8
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