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Discovery of Oral Natural Benzofuranoid p -Terphenyl Derivative CHNQD-03301 as a Potent Hypoxia-Inducible Factor-1α Signaling Inhibitor for Cancer Therapy

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Year: 2025
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.5c01859
Authors: Cui-Fang Wang, Xiao-Nan Cui, Liu-Xia Lv, Wen-Hui Wang, Qian-Qian Jing, Jun-Na Yin, Xi-Zhen Cao, Mei-Yan Wei, Ling Lu, Chang-Lun Shao
Institutions: Ministry of Education of the People's Republic of China, Ocean University of China, Qingdao National Laboratory for Marine Science and Technology
Language: English

Topic: Cancer, Hypoxia, and Metabolism
Subfield: Cancer Research
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: National Natural Science Foundation of China, Qingdao National Laboratory for Marine Science and Technology, State Key Laboratory for Chemistry and Molecular Engineering of Medicinal Resources
Awards: G1099348271, G2886852188, G6054668379, G616954693, G7306024628, G7791230303
OpenAlex ID: W4415656198
FWCI: 0.337
Cites: 41
Cited by: 1
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