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Discovery and Characterization of VPRBP/DCAF1 Kinase Inhibitor Analogs as Microtubular Destabilizing Agents with Potent Antimyeloma Activity

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Year: 2025
Type: article
Source: Molecular Cancer Therapeutics
DOI: 10.1158/1535-7163.mct-25-0306
Authors: Olivia Susanto, Emily Gruber, Cheng Mun Wun, Rheana L. Franich, Xiao Ma, Zahra Sabouri-Thompson, Zoe J. Porter, Heather C. Murray, Leonie A. Cluse, Belinda Maher, Daniella Brasacchio, Benjamin P. Martin, Peter J. Fraser, Iva Nikolic, Gisela Mir Arnau, Jarrod J. Sandow, Kaylene J. Simpson, Nicole M. Verrills, Ricky W. Johnstone, Philip E. Thompson, Lev M. Kats, Jake Shortt
Institutions: Monash Health, Monash University, The University of Melbourne, Peter MacCallum Cancer Centre, Hunter Medical Research Institute, University of Newcastle Australia, Monash Medical Centre, Victorian Centre for Functional Genomics, Vall d'Hebron Institute of Oncology, Walter and Eliza Hall Institute of Medical Research
Language: English

Topic: Multiple Myeloma Research and Treatments
Subfield: Hematology
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: Leukemia and Lymphoma Society, Leukaemia Foundation, Cancer Council Victoria
Award: G906436120
OpenAlex ID: W4415846858
FWCI: 0.638
Cites: 58
Cited by: 1
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