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Discovery and Optimization of a Non-Nucleoside-Based Series of Inhibitors of 2′-Deoxynucleoside 5′-Monophosphate Glycosidase (DNPH1)

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Year: 2025
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.5c02356
Authors: Bernard Barlaam, Luz Alonso-Crisostomo, Niall A. Anderson, Argyrides Argyrou, Peter C. Astles, Elaine B. Cadogan, Luca Carlino, Gavin W. Collie, Nichola L. Davies, James Hall, Linda Kitching, Xianxi Li, Filippos Michopoulos, Alexander G. Milbradt, Jenni Nikkilä, Sarah Northall, Mark J. O’Connor, Xiaohiu Pei, Joseph Shaw, Danial Slade, Harriet Southgate, Darren Stead, Christopher J. Stubbs, Benjamin C. Whitehurst, Bin Xing, Yihao Yuan, Jie Zhou
Institutions: AstraZeneca (United Kingdom), Pharmaron (China)
Language: English

Topic: PARP inhibition in cancer therapy
Subfield: Oncology
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W4415950120
FWCI: 0.362
Cites: 13
Cited by: 1
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