Major Progress in the Liquid-Phase Synthesis of N -Alkyl-Rich Cyclic Peptides: Kilogram-Scale GMP Production of the KRAS Inhibitor LUNA18
Year: 2025
Type: article
Authors: Zengye Hou, Shio Komiya, Kotaro Iwasaki, Yasuhiro Kondo, Yousuke Momose, Kiyoshi Sasakura, Kota Tanaka, Manabu Wadamoto, Peithing Chia, Katsunori Dan, Hirotaka Ejima, Hiroki Fujisawa, Akira Fukuzawa, Shohei Hashimoto, Takenori Ishizawa, Hisashi Ito, Yuki Nakagawa, Hitomi Sato, Nao Sato, Hiroko Sekita, Hiroki Serizawa, Sayako Tamura, Taro Enomoto, Akie Honma, Takuma Ikeda, Masatoshi Murakata, Junichi Shiina, Takahiko Yabuzaki, Masao Tsukazaki, Hiroshi Iwamura, Kenji Maeda
Institution: Chugai Pharmaceutical Co., Ltd. (Japan)
Language: English
Subfield: Molecular Biology
Domain: Life Sciences
Open Access status: closed
OpenAlex ID: W4416109532
