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Discovery and Characterization of Novel BLIMP-1 Heterobifunctional Ligand-Directed Degraders

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Year: 2025
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.5c02363
Authors: Bryan J. Simmons, Lynda Groocock, Jesus Moreno, David S. Peters, Meredith E. Hughes, Vijay Veeravalli, Jennifer M. Crawford, Matthew Chalkley, Mark Griffith, Melissa Plooster, Bo Hu, Jim Gamez, Jim Leisten, Michael J. Barnes, Jason Chinn, Gauri Deb, Hardik Modi, Madhu Katepalli, Dahlia Weiss, Walter Won, Zhenghang Sun, Shan Yu, Cameron Reid, Andrew F. Donnell, Ling Li, Edmond R. Watson, Sophie Perrin-Ninkovic, Lihong Shi, Rama Krishna Narla, Christoph W. Zapf, Neil Bence, Antonia Lopez-Girona, Jennifer R. Riggs
Institutions: Bristol-Myers Squibb (United States), Bristol-Myers Squibb (United Kingdom)
Language: English

Topic: Protein Degradation and Inhibitors
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W4416584994
FWCI: 0.253
Cites: 18
Cited by: 1
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