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Targeting Chikungunya virus entry: Enantiomeric separation, synthesis of derivatives, and structure-activity relationship of E1-E2 envelope glycoprotein inhibitors

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Year: 2025
Type: article
Source: European Journal of Medicinal Chemistry
DOI: 10.1016/j.ejmech.2025.118427
Authors: Daniela M. Fidalgo, Eliana Castro, Agostina Mazzeo, Tamara J.B. Vazquez, Leandro Battini, Daniel Vladimir, Malena Tejerina Cibello, Facundo N. Gallo, Maximilian A. Rey, Sara A. Thannickal, Sophie N. Spector, Florencia Di Salvo, María E. Monge, Kenneth A. Stapleford, Diego E. Alvarez, Mariela Bollini
Institutions: Consejo Nacional de Investigaciones Científicas y Técnicas, National University of General San Martín, Universidad de Buenos Aires, New York University, Instituto de Química-Física de los Materiales, Medio Ambiente y Energía
Language: English

Topic: Mosquito-borne diseases and control
Subfield: Public Health, Environmental and Occupational Health
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: Consejo Nacional de Investigaciones Científicas y Técnicas, Cambridge Crystallographic Data Centre, Agencia Nacional de Promoción Científica y Tecnológica
Awards: G455821934, G742075266
OpenAlex ID: W4416828694
FWCI:
Cites: 22
Cited by:
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