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Discovery, Design, and Synthesis of Novel 2-Benzyl-2,7-diazaspiro[3.5]nonane Benzothiazinones with Broad-Spectrum Antimycobacterial Activity

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Year: 2025
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.5c02429
Authors: Jizhou Wu, Chao Ma, Meng Wei, Xiuzhen Chen, Weixiao Wang, Jinghan Gao, Junjie Huang, Xiaorui Ji, Meijiao Wei, Mingliang Liu, Apeng Wang, Kai Lv, Wei Chen
Institutions: Chinese Academy of Medical Sciences & Peking Union Medical College, Nanjing University of Chinese Medicine
Language: English

Topic: Phenothiazines and Benzothiazines Synthesis and Activities
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: National Natural Science Foundation of China, Chinese Academy of Medical Sciences, Nanjing Municipal Health Bureau, Beijing Municipal Natural Science Foundation
Awards: G1503162417, G2678509557, G4139562353, G5153934310, G7917612554
OpenAlex ID: W4417259686
FWCI: 0.261
Cites: 29
Cited by: 1
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