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Table S4 from PRT3789 Is a First-in-Human SMARCA2-Selective Degrader That Induces Synthetic Lethality in SMARCA4-Mutated Cancers

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Year: 2026
Type: other
Abstract: IC50 Values of PRT3789 for Anti-Proliferation in Various Tumor Cell Lines in 2D In Vitro Assay
DOI: 10.1158/0008-5472.30985998
Authors: Michael Hulse, Min Wang, Chaoyi Xu, Jack Carter, Anjana Agarwal, Liang Lu, Philip Pitis, Neha Bhagwat, Joseph Rager, Justin Kurian, Corey Basch, Monisha Sivakumar, Jessica Burtell, Arpita Mondal, Alexander Grego, Andrew Moore, Carly Bachner, Komali Vykuntam, Anthony Reichelderfer, Jimin Park, Joy Cote, Miles Cowart, Olusola Peace Osinubi, Ludovic Bigot, Alice Da Silva, Catline Nobre, Melissandre Meteau, Miguel Soares, Hsin-Yao Tang, Klare Bersch, Chaofeng Dai, Ganfeng Cao, Bo Shen, Tom Emm, Stefan Ruepp, Jennifer Xavier, Chris Tankersley, Diane Heiser, Sang Hyun Lee, Sandy Geeganage, Bruce Ruggeri, Hong Lin, William Novotny, Jane Huang, Kris Vaddi, Andrew Combs, Peggy Scherle, Koichi Ito
Language: English

Topic: Protein Degradation and Inhibitors
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: gold
OpenAlex ID: W7117968510
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Related to: 10
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