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Discovery of AZD9750, an Orally Bioavailable Androgen Receptor Degrader for the Treatment of Prostate Cancer

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Year: 2026
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.5c03138
Authors: James S. Scott, Laura Evans, Peter C. Astles, Argyrides Argyrou, Sharan K. Bagal, David Beattie, Erin L. Braybrooke, Doyle J. Cassar, Claire Crafter, Coura Diène, Gary Fairley, Charlene Fallan, Graham Fraser, Nuria Galeano-Dalmau, Thomas G. Hammond, Andreas K. Hock, Thomas Jones, Jasper Komen, Gillian M. Lamont, Chrysiis Michaloglou, Michael J. Niedbala, Antonio Ramos-Montoya, Monica C. Rodrigo-Brenni, Martin J. Packer, Stuart Pearson, Andy Pike, Markus Schade, Joseph Shaw, Ziyanda Shologu, Oliver Steward
Language: English

Topic: Protein Degradation and Inhibitors
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funder: AstraZeneca
OpenAlex ID: W7126262948
FWCI: 12.75
Cites: 35
Cited by: 7
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