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[ 68 Ga]Ga-PG2-2FAPI: A DPro-Gly-Modified Dimeric FAPI Probe with Enhanced Tumor Uptake and Retention

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Year: 2026
Type: article
Source: Molecular Pharmaceutics
DOI: 10.1021/acs.molpharmaceut.5c01824
Authors: Qing Ruan, Yuhao Jiang, Zuojie Li, Xiaojiang Duan, Lina Diao, Dajie Ding, Peiwen Han, Guangxing Yin, Jianyong Jiang, Junbo Zhang
Institutions: National Medical Products Administration, Beijing Normal University, Ministry of Education, Peking University First Hospital
Language: English

Topic: Peptidase Inhibition and Analysis
Subfield: Oncology
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: National Natural Science Foundation of China, Beijing Municipal Natural Science Foundation, Beijing Nova Program, Fundamental Research Funds for the Central Universities
Awards: G2453141964, 靶向细菌性感染的放射性核素标记抗菌肽衍生物的制备和显像研究, G6534191486, G716361101, 靶向PSMA的99mTc标记含三唑环的谷氨酸-脲衍生物用作肿瘤分子探针的研究, G757220836
OpenAlex ID: W7128036146
FWCI: 2.68
Cites: 31
Cited by: 1
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