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Design, synthesis and biological evaluation of Rac1-targeting carbazole–pyrimidines as host-directed antimalarials

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Year: 2026
Type: article
Source: European Journal of Medicinal Chemistry
DOI: 10.1016/j.ejmech.2026.118690
Authors: Silvia Parapini, Sarah D'Alessandro, Sara Travaglione, Silvio Paone, Ileanexis M. Madera Cuevas, Teresa Dipol, Davy Wendyam Raoul Zongo, Ana M. Figueroa Vázquez, Ornella Morsilli, Alessia Fabbri, Cornelis P. Vlaar, Anna Olivieri
Institutions: University of Milan, Istituto Superiore di Sanità, University of Puerto Rico, Medical Sciences Campus, University of Puerto Rico System, Sapienza University of Rome
Language: English

Topic: Malaria Research and Control
Subfield: Public Health, Environmental and Occupational Health
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: Istituto Superiore di Sanità, Puerto Rico Science, Technology and Research Trust
OpenAlex ID: W7129097819
FWCI: 6.375
Cites: 43
Cited by: 1
Related to: 10
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