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The Use of Glycine-Containing Peptide-Based Chelators for Labeling with 99m Tc Improves the Imaging Properties of EpCAM-Targeting Designed Ankyrin Repeat Ec1

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Year: 2026
Type: article
Source: Molecular Pharmaceutics
DOI: 10.1021/acs.molpharmaceut.5c01498
Authors: Sergey Deyev, Anastasia Fominykh, Ruslan Varvashenya, Gleb Yanovich, Vitalina Bodenko, Evgenii Plotnikov, Mariia Tretyakova, Daria Eskova, Roman Zhelchan, Alexey Schulga, Elena Konovalova, Rustam Ziganshin, Anna Orlova, Mikhail Belousov, Vladimir Tolmachev, Mariia Larkina
Institutions: Russian Academy of Sciences, Tomsk Polytechnic University, Institute of Bioorganic Chemistry, Tomsk National Research Medical Center, Tomsk Cancer Research Institute, Institute of Bioorganic Chemistry, Uppsala University, Siberian State Medical University
Language: English

Topic: Radiopharmaceutical Chemistry and Applications
Subfield: Radiology, Nuclear Medicine and Imaging
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funder: Tomsk Polytechnic University
Award: G1832087533
OpenAlex ID: W7133521152
FWCI: 9.045
Cites: 47
Cited by: 2
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