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Discovery of Non-prostanoid EP4 Agonists for the Treatment of Inflammatory Bowel Disease

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Year: 2026
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.6c00130
Authors: Heidi L. Perez, Sunita Dewnani, Steven A. Spronk, Hai-Yun Xiao, Ling Li, Mojgan Abousleiman, Chi Shing Sum, Margarita Garcia-Calvo, Fei Yu, Brian Anderson, Brian J. Arey, Riyaz Khan, Chandra Sekhar Bokka, Yazh Muthukumar, Kaushik Ghosh, Tao Wang, Carol M. Krause, Judith Murray, Trevor Vernon, Ramakrishna Chandran, Mary T. Obermeier, Victor R. Guarino, Tamara King, Julia Li, Laura Armstrong, Purnima Khandelwal, Margaret Prack, David Marcoux, Samuel Gerritz, William J. Pitts, Alaric J. Dyckman, Robert M. Borzilleri, Carolyn Dzierba, Jenny H. Xie, Mary Struthers, Patrick Shaw, Derek Holmes, Amy C. Hart, Trevor C. Sherwood
Institutions: Bristol-Myers Squibb (United States), Bristol-Myers Squibb (United Kingdom)
Language: English

Topic: Inflammatory mediators and NSAID effects
Subfield: Pharmacology
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W7148653479
FWCI:
Cites: 25
Cited by:
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