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Abstract 6734: Discovery and optimization of NEO-811, a first-in-class molecular glue degrader of ARNT, utilizing structure-based drug design.

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Year: 2026
Type: conference-abstract
Source: Cancer Research
DOI: 10.1158/1538-7445.am2026-6734
Authors: Jennifer Griffin, Andres Hernandez, Xiaoxi Liu, Kurt Januszyk, Bryan Lee, Anthony Burt, John Tellew, J. Scott Lee, Michelle Cruz, Isabella Tran, Kevin Chiu, Mengyu Wu, Leslie Bateman, Ana Dominguez-Andres, Ling Huang, Jake Fathman, Celin Sanchez, Nathalia Cruz, Randy Soriano, Devin Knece, Molly Fitzgibbon, Ana Grant, Mary Matyskiela, Rohan Beckwith, Phil Chamberlain
Institution: Neomorph
Language: English

Topic: Protein Degradation and Inhibitors
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W7148846753
Cites:
Cited by: 1
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