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Discovery of INCB191358: A Potent and Selective DGKα/ζ Dual Inhibitor

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Year: 2026
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.5c03768
Authors: Bo Wei, Xiaolei Li, Jacob J. Lacharity, Liana Hie, Dingquan Qian, Melissa Chan, David Rodrigues, Kelly Federowicz, Guofeng Zhang, Gengjie Yang, Maryanne Covington, Bihui Melidosian, Jeff Jackson, Lisa Truong, Michelle Frascella, Xiaodi Ren, Rodrigo Hess, Patrick Mayes, Sunkyu Kim, Joshua R. Hummel, Xiaozhao Wang
Institution: Incyte (United States)
Language: English

Topic: Protein Kinase Regulation and GTPase Signaling
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funder: Incyte
OpenAlex ID: W7154686986
FWCI:
Cites: 68
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