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Rational Design, Synthesis, and Biological Evaluation of Potent, Highly Selective 1,2,4-Oxadiazole-Based S1PR1 Agonists for UC Treatment

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Year: 2026
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.5c03837
Authors: Tianyu Ye, Yunping Xiao, Chenyang Tang, Jinling Yu, Luqi Zhang, Zhongping Xu, Simeng Huang, Ranran Wang, Ranran Wang, Shengliang Jin, Zhenjiang Zhao, Huan He, Rui Wang, Rui Wang, Lili Zhu, Honglin Li
Institutions: East China University of Science and Technology, East China Normal University
Language: English

Topic: Sphingolipid Metabolism and Signaling
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: National Natural Science Foundation of China, National Key Research and Development Program of China
Awards: G1618279006, G5009833721, G5524584715
OpenAlex ID: W7154739307
FWCI:
Cites: 68
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