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Discovery of CN-3 as a Next-Generation RET Inhibitor Potently Overcoming Multiple Mutations

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Year: 2026
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.6c00376
Authors: Zi-Xuan Wang, Rui He, Min-Hui Chen, Kun Yang, Qian Liu, Jin Yang, Meng-Yuan Zhang, Nuo Qiao, Ming-Dan Zhou, Yan-Cheng Yu, Shan-Liang Sun, Yuan-Hui Lai, Ye Yang, Zhang Zhang, Nian-Guang Li, Zhi-Hao Shi
Institutions: Nanjing University of Chinese Medicine, Jinan University, China Pharmaceutical University
Language: English

Topic: Lung Cancer Treatments and Mutations
Subfield: Pulmonary and Respiratory Medicine
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: National Natural Science Foundation of China, Nanjing University of Chinese Medicine
Awards: G3270552589, G5191291281, G5913327515, G6771631603
OpenAlex ID: W7159953586
FWCI:
Cites: 43
Cited by:
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