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Discovery of Fosigotifator, a Potent eIF2B Activator with Desired Properties for Human Studies

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Year: 2026
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.6c00716
Authors: Jennifer M. Frost, Yunsong Tong, Xiangdong Xu, Lei Shi, Marina Pliushchev, Kathleen J. Murauski, Kathy Kohlhaas, Diana L. Donnelly-Roberts, Michael M. Sheehan, Stephan Riedmaier, Hardeep S. Oberoi, Jun Chen, Janani Prakash, Charles W. Hutchins, Clarissa G. Jakob, Rinku Jain, Wei Qiu, Rodger F. Henry, Rohinton Edalji, Chaohong Sun, Tracy Carr, Ana M. Basso, Brian S. Brown, Eric A. Voight, Carmela Sidrauski, Michael J. Dart
Institution: Calico Life Sciences
Language: English

Topic: Endoplasmic Reticulum Stress and Disease
Subfield: Cell Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: AbbVie, Calico Life Sciences
OpenAlex ID: W7161633049
FWCI: 9.187
Cites: 33
Cited by: 3
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