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Discovery of Dual A2A/A2B Adenosine Receptor Antagonist and Clinical Candidate INCB106385

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Year: 2026
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.6c00964
Authors: Chao Qi, Matthew S. McCammant, Yong Li, Wenyu Zhu, Zhiyong Yu, Peter Carlsen, Heeoon Han, Le Zhao, Fenglei Zhang, Taisheng Huang, Pei Gan, Dingquan Qian, Gia Hoang, Chunhong He, Song Mei, Jennifer J. Harris, Alexandra Gallion, Michael Hansbury, Jennifer Mason, Kristine Stump, Kerri Kurzeja-Lipinski, Angela DiRamio, Maryanne Covington, Holly Koblish, Sharon Diamond, Hui Wang, Peggy Scherle, Wenqing Yao, Xiaozhao Wang
Institution: Incyte (United States)
Language: English

Topic: Adenosine and Purinergic Signaling
Subfield: Physiology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funder: Incyte
OpenAlex ID: W7162490259
FWCI:
Cites: 39
Cited by:
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