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Lysine-Targeted Covalent Inhibitors: Emerging Warheads and Expanding Applications in Medicinal Chemistry

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Year: 2026
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.5c03241
Authors: Yue Wu, Yafen Chen, Ruiheng Cao, Xiang Li, Xiaojin Zhang
Institution: China Pharmaceutical University
Language: English

Topic: Click Chemistry and Applications
Subfield: Organic Chemistry
Field: Chemistry
Domain: Physical Sciences

Open Access status: closed

Funders: National Natural Science Foundation of China, China Postdoctoral Science Foundation, Basic Research Program of Jiangsu Province, Fundamental Research Funds for the Central Universities
Awards: G1481093169, G2376736480, G3005621743, G4311388668, G5001627880, G5424221654, G6411985011, G7140215128, G917615550
OpenAlex ID: W7162512969
FWCI: 5.402
Cites: 112
Cited by: 3
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