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Phase I/IIa study of DN022150, a novel selective noncovalent small molecule KRAS G12D inhibitor in patients with advanced KRAS G12D–mutant solid tumors.

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Year: 2026
Type: conference-abstract
Source: Journal of Clinical Oncology
DOI: 10.1200/jco.2026.44.16_suppl.3007
Authors: Yiyi Yu, Tianshu Liu, Junli Xue, Wei Zhao, Yuping Sun, Xudong Hu, Shuqin Ni, Yuejuan Cheng, Yuan Liu, Ting Deng, Zhi Ji, Yongchang Zhang, Xue Chen, Jing Sun, Ting Wang, Xicheng Wang, Qiongfei Su, Xiao Chen, Haiwei Fan, Shousheng Yan
Institutions: Fudan University, Zhongshan Hospital, Shanghai East Hospital, Shandong Tumor Hospital, Peking Union Medical College Hospital, Tianjin Medical University Cancer Institute and Hospital, Tianjin Medical University, Hunan Cancer Hospital, Jiangsu Province Hospital, Guangdong Pharmaceutical University, First Affiliated Hospital of Guangdong Pharmaceutical University
Language: English

Topic: Protein Kinase Regulation and GTPase Signaling
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W7162556914
Cites:
Cited by: 2
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