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Structure-Guided Designed [18F]-labeled FAPI for Enhanced Hydrophilicity: From Preclinical to First-In-Human Study

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Year: 2026
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.5c03486
Authors: Xingyu Mu, Lei Zhang, Zihao Chen, Hoi Yee Chow, Jingze Li, Weixia Chong, Yufeng Mo, Ganghua Tang, Xuechen Li, Wei Fu
Institutions: Guilin Medical University, Southern Medical University, University of Hong Kong
Language: English

Topic: Radiopharmaceutical Chemistry and Applications
Subfield: Radiology, Nuclear Medicine and Imaging
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: Natural Science Foundation of Guangxi Zhuang Autonomous Region, Morningside Foundation, National Natural Science Foundation of China, Guangxi Zhuang Autonomous Region Health and Family Planning Commission
Awards: G1951911628, G3056884511, G3243413948, G8012808915
OpenAlex ID: W7162784293
FWCI: 13.57
Cites: 36
Cited by: 3
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