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Design, Synthesis, and Evaluation of [ 68 Ga/ 177 Lu]-Labeled TSPO-Targeting Radioligands for PET/CT Diagnosis and Radionuclide Therapy of Brain Tumor

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Year: 2026
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.5c03527
Authors: Xingkai Wang, Siqi Zhang, Yiming Li, Can Liu, Jiang Wu, Yuxuan Wu, Qichen Hu, Wenhao Liu, Qingshuang Lu, Xindan Hu, Dong Dai, Yingzi Zhang, Zhong Zhang, Feng Wang, Rui Wang, Kuan Hu
Institutions: Chinese Academy of Medical Sciences & Peking Union Medical College, Tianjin Medical University Cancer Institute and Hospital, Capital Medical University, Beijing Tian Tan Hospital, Nanjing First Hospital, Nanjing Medical University, Second Affiliated Hospital of Soochow University
Language: English

Topic: Radiopharmaceutical Chemistry and Applications
Subfield: Radiology, Nuclear Medicine and Imaging
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funder: National Natural Science Foundation of China
Awards: G1863677309, G4969500791
OpenAlex ID: W7164989656
FWCI: 4.555
Cites: 70
Cited by: 1
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