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Unique Cysteine-Directed Covalent Inhibition of PRMT1 Suppresses Breast Tumorigenesis

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Year: 2026
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.6c00262
Authors: Min Shao, Ruining Li, Jinglei Hu, Wenjie Xi, Raghupathi Mutyala, Lulu Guan, Chaoqun Huang, Renhong Sun, Xiaobao Yang, Bo Jin, Bo Zhao, Erjun Hao, Zhimin Zhang, Lin Li, Xufen Yu, Mingyan Zhu, Yudao Shen
Institutions: Shanghai Jiao Tong University, Henan Normal University, Fudan University, Key Laboratory of Smart Drug Delivery, Ministry of Education, Jinan University, Central Research Institute
Language: English

Topic: Cancer-related gene regulation
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: Natural Science Foundation of Henan Province, National Key Research and Development Program of China
Awards: G5564223311, G7935452240, G943023285
OpenAlex ID: W7164998186
FWCI:
Cites: 55
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