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A Review of Population Pharmacokinetic Models and Dosing Algorithms Assessing the Influence of CYP3A5 Genotype and Other Clinical Covariates on Tacrolimus Pharmacokinetics

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Year: 2026
Type: article
Source: Clinical Pharmacokinetics
DOI: 10.1007/s40262-026-01673-x
Authors: Riley M. Randolph, Sara Jubas, Li Gong, Raman Venkataramanan, Dhrita Khatri, Pamala A. Jacobson, David Metz, Daniel J. Crona
Institutions: University of North Carolina at Chapel Hill, Stanford University, University of Pittsburgh, The University of Melbourne, Murdoch Children's Research Institute, University of Minnesota, Royal Children's Hospital, Monash Children’s Hospital, Monash Health, Monash University, UNC Lineberger Comprehensive Cancer Center
Language: English

Topic: Pharmacogenetics and Drug Metabolism
Subfield: Pharmacology
Field: Pharmacology, Toxicology and Pharmaceutics
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: National Human Genome Research Institute, National Institute of General Medical Sciences, Medical Research Future Fund
Awards: G1078340221, G738042423, Minimising Adverse drug Reactions and Verifying Economic Legitimacy - Pharmacogenomics Implementation in Children (MARVEL-PIC), Clinical Implementation Resources for Pharmacogenomics (CIRP)
OpenAlex ID: W7169774665
FWCI:
Cites: 143
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