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Abstract B047: dCBP-30: A rationally designed, orally bioavailable, near-linkerless PROTAC for potent CBP/p300 degradation

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Year: 2026
Type: conference-abstract
Source: Clinical Cancer Research
DOI: 10.1158/1557-3265.d32026-b047
Authors: Praveen Kumar. Tiwari, Bomin Ku, Sai Reddy. Doda, Drew A. Harrison, Sarah Rizvi, Samuel Ojeda, Jessica Jessica Duffy, Leonie Cluse, Jennifer R. Devlin, Nenad Bartonicek, Olga Motorna, Ann-Sophie Koglin, Barbara Karakyriakou, Kaitlyn Gagnon, Ramya S. Iyer, Regina Egan, Pat Greninger, Lauren Benz, Caroline Greco, Julia Norton, Amruth Kumar, Eric F. Zaniewski, Soroush Hajizadeh, Robert Morris, Genna Mullen, Ajinkya S. Kawale, Sangwon Min, Raghu Vannam, Lee Zou, Wilhelm Haas, Abner Louissaint, Ricky W. Johnstone, Christopher J. Ott
Institutions: Harvard University, Massachusetts General Hospital, The University of Melbourne, Peter MacCallum Cancer Centre
Language: English

Topic: Protein Degradation and Inhibitors
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W7169857430
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