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BE2012 a novel, REV-ERB antagonist that promotes regenerative myogenesis in vivo with substantially improved pharmacokinetics relative to SR8278

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Year: 2026
Type: article
Source: Journal of Pharmacology and Experimental Therapeutics
DOI: 10.1016/j.jpet.2026.105011
Authors: Isabelle Cote, Aurore C. Valfort, Ryan K. Sanders, Sheryl L. Burris, Matthew E. Hayes, Rhea Arya, Lingaiah Maram, Bahaa Elgendy, Feng Yue, Thomas P. Burris
Institutions: University of Florida, University of Health Sciences and Pharmacy, Washington University in St. Louis, Institute of Food and Agricultural Sciences
Language: English

Topic: Muscle Physiology and Disorders
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funder: Sucampo Pharmaceuticals
OpenAlex ID: W7203622517
FWCI:
Cites: 32
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