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Optimization of a Series of Novel 1 H -Pyrrolo[3,2- c ]pyridine-Based USP1 Inhibitors with Potent In Vivo Antitumor Activity

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Year: 2026
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.6c01009
Authors: Tao Yang, Xue Cui, Qingyan Li, Yaxin Teng, Minghai Tang, Xinyu Zou, Xiaobo Cen, Lijuan Chen, Min Zhao, Linyu Yang, Zhuang Yang
Institution: Sichuan University
Language: English

Topic: Ubiquitin and proteasome pathways
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: National Natural Science Foundation of China, Natural Science Foundation of Sichuan Province, West China Hospital, Sichuan University
Awards: G4686701503, G6047992252, G7148227395, G7522400348
OpenAlex ID: W7203706683
FWCI:
Cites: 39
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