Work

Dual‐Site Covalent Targeting Enables BD2‐Selective BET Inhibition With Potent Antitumor Activity in Mice

Year: 2026

Type: article

Source: Angewandte Chemie

DOI: 10.1002/ange.1224416

Authors: Jibo Kang, Xuan Wang, Hong Zhang, Jieying Lin, Peng Chen, Zuqin Wang, Zengjun Hao, Fengfei Miao, Fengcai Zhang, Tao Li, Yusheng Xie, Junjian Wang, Zhi‐Min Zhang, Shao Q. Yao, Xiaoyun Lu

Institutions: Jinan University, National University of Singapore, Shandong University, Sun Yat-sen University

Language: English

Topic: Protein Degradation and Inhibitors

Subfield: Molecular Biology

Field: Biochemistry, Genetics and Molecular Biology

Domain: Life Sciences

SDG: Good health and well-being

Open Access status: closed

Funders: National Natural Science Foundation of China, National Medical Research Council, National Key Research and Development Program of China

Awards: G1827903050, G4646048394, G7126553680, G7756859128

OpenAlex ID: W7208716503

FWCI:

Cites: 27

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