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From Inhibitor to Reporter: Nirmatrelvir-Derived Fluorogenic Substrates for the SARS-CoV-2 Main Protease

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Year: 2026
Type: article
Source: ACS Chemical Biology
DOI: 10.1021/acschembio.6c00577
Authors: Rabea Voget, Victoria Steiger, Katharina Sylvester, Chun-Chiao Yang, Louisa von Kohout, Dominik Thimm, Julian Breidenbach, Norbert Sträter, Christa E. Müller, Michael Gütschow
Institutions: University of Bonn, Leipzig University
Language: English

Topic: SARS-CoV-2 and COVID-19 Research
Subfield: Infectious Diseases
Field: Medicine
Domain: Health Sciences

Open Access status: closed

Funders: Deutsche Forschungsgemeinschaft, Volkswagen Foundation
Awards: G27865616, GRK 2873: Werkzeuge und Wirkstoffe der Zukunft Innovative Methoden und neue Modalitäten in der Medizinischen Chemie, G6943711111
OpenAlex ID: W7208816534
FWCI:
Cites: 57
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