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Structure-Guided Design, Synthesis, and Evaluation of Novel 6-Methoxyquinoline-4-carboxamide Derivatives as First-in-Class Nano-Molar B3GAT3 Inhibitors for the Treatment of Hepatocellular Carcinoma

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Year: 2026
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.6c02080
Authors: Hao Yin, Xiaowen Yan, Bo Fan, Xiangye Kong, Congying Gu, Wang Zhou, Shiping Xu, Zenglin Yin, Min Zhang, Youchen Wang, Hongyan Liu, Junli Feng, Lei Ge, Jiacheng Li, Tangtai Dong, Yong Yang, Dayong Zhang, Beiying Dai, Menghan Zhang
Institution: China Pharmaceutical University
Language: English

Topic: Synthesis and biological activity
Subfield: Organic Chemistry
Field: Chemistry
Domain: Physical Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: China Pharmaceutical University, Natural Science Foundation of Jiangsu Province, State Key Laboratory of Natural Medicines
Awards: G2755637204, G6873476444, G7377214975, G8447373577
OpenAlex ID: W7212289670
FWCI:
Cites: 45
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