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Restoration of PP2A AαB56αC trimer formation by RPT04402 molecular glue in high-grade uterine cancer

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Year: 2026
Type: article
Source: Science Translational Medicine
DOI: 10.1126/scitranslmed.ady4852
Authors: Irene Peris, Terrance J. Haanen, Alexander Day, Jiang Hu, Catherine Callahan, Gabrielle Hodges-Onishi, Kaitlin P. Zawacki, Brian Tran, Alexis Harold, Amanda Dowdican, Charles A. Nino, Wei Huang, Daniel Leonard, Matthew Hinderman, Kelsey Barrie, Brynne Raines, Jaya Sangodkar, Sophie Boock, Varsha Shankar, Miranda Giambi, Silvia Romero-Murillo, Leah Arbitman, Shirish Shenolikar, George Trainor, Frederic Cachoux, Obdulia Rabal, Olga Gherbovet, Laura Fourmois, David L. Brautigan, Analisa V. DiFeo, Derek J. Taylor, Caitlin M. O’Connor, Goutham Narla
Institutions: University of Michigan, Michigan Medicine, Michigan Cancer Research Consortium, Case Western Reserve University, Universidad de Navarra, Signature Research (United States), Evotec (United States), University of Virginia
Language: English

Topic: Protein Degradation and Inhibitors
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: U.S. Department of Defense, National Institutes of Health, National Cancer Institute
Awards: G1686049839, G4390880649, G9001196726, G9001204161, G9001227182
OpenAlex ID: W7221806993
FWCI:
Cites: 41
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