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Methadone: Historical success, modern challenges and lessons for opioid drug discovery

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Year: 2026
Type: review
Source: Drug Discovery Today
DOI: 10.1016/j.drudis.2026.104840
Authors: Ennian Li, Preet Shah, Yan Zhang
Institution: Virginia Commonwealth University
Language: English

Topic: Pain Management and Opioid Use
Subfield: Anesthesiology and Pain Medicine
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: green

Funder: National Institute on Drug Abuse
Awards: Development of Specific Mu Opioid Receptor Antagonists to Reverse the Acute and Chronic Toxicity of Fentanyls, Mu Opioid Receptor Modulator Development to Treat Opioid Use Disorder, Mu Opioid Receptor Modulator Development to Treat Opioid Use Disorder
OpenAlex ID: W7223325990
FWCI:
Cites: 74
Cited by:
Related to: 10
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