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Enthalpy-Informed Design of Dasatinib-Derived Small-Molecule Inhibitors of Transthyretin Amyloidogenesis

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Year: 2026
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.6c02395
Authors: Takeshi Yokoyama, Airi Fukugawa, Ryoka Waki, Katsuhiro Kusaka, Haruki Sugiyama, Yuko Nabeshima, Mineyuki Mizuguchi, Takuya Okada, Naoki Toyooka
Institutions: University of Toyama, Comprehensive Research Organization for Science and Society
Language: English

Topic: Amyloidosis: Diagnosis, Treatment, Outcomes
Subfield: Internal Medicine
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funder: Japan Society for the Promotion of Science
OpenAlex ID: W7225454932
FWCI:
Cites: 34
Cited by:
Related to: 10
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