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Michael H. Rabinowitz
Observed names:
M Rabinowitz,
M. H. RABINOWITZ,
Michael H Rabinowitz,
Michael Rabinowitz,
Rabinowitz, M.H.,
Rabinowitz, Michael
show all 6
Institution:
Akebia Therapeutics (United States)
Observed institutions:
University of California, Irvine,
Akebia Therapeutics (United States),
GlaxoSmithKline (United States),
Wallace Laboratories,
Janssen Research & Development (United States),
Stanford University
show all 6
OpenAlex ID:
A5000389847
Enantioselective Total Synthesis of (-)-Ptilomycalin A
1995
·
Larry E. Overman
, Michael H. Rabinowitz
, et al.
·
Journal of the American Chemical Society
·
210
Inhibition of Hypoxia-Inducible Factor Prolyl Hydroxylase Domain Oxygen Sensors: Tricking the Body into Mounting Orchestrated Survival and Repair Responses
2013
·
Michael H. Rabinowitz
·
Journal of Medicinal Chemistry
·
165
The first enantioselective total syntheses of the allopumiliotoxin A alkaloids 267A and 339B
1992
·
Steven W. Goldstein
, Larry E. Overman
, et al.
·
The Journal of Organic Chemistry
·
85
Inhibition of Tumor Necrosis Factor-α (TNF-α) Production and Arthritis in the Rat by GW3333, a Dual Inhibitor of TNF-α-Converting Enzyme and Matrix Metalloproteinases
2001
·
James G. Conway
, Robert C. Andrews
, et al.
·
Journal of Pharmacology and Experimental Therapeutics
·
82
Pharmacological Characterization of 1-(5-Chloro-6-(trifluoromethoxy)-1H-benzoimidazol-2-yl)-1H-pyrazole-4-carboxylic Acid (JNJ-42041935), a Potent and Selective Hypoxia-Inducible Factor Prolyl Hydroxylase Inhibitor
2011
·
Terrance D. Barrett
, Heather L. Palomino
, et al.
·
Molecular Pharmacology
·
80
Design of Selective and Soluble Inhibitors of Tumor Necrosis Factor-α Converting Enzyme (TACE)
2001
·
Michael H. Rabinowitz
, Robert C. Andrews
, et al.
·
Journal of Medicinal Chemistry
·
73
A Practical Entry to the Crambescidin Family of Guanidine Alkaloids. Enantioselective Total Syntheses of Ptilomycalin A, Crambescidin 657 and Its Methyl Ester (Neofolitispates 2), and Crambescidin 800
2000
·
D. Scott Coffey
, Andrew I. McDonald
, et al.
·
Journal of the American Chemical Society
·
66
Benzimidazole-2-pyrazole HIF Prolyl 4-Hydroxylase Inhibitors as Oral Erythropoietin Secretagogues
2010
·
Mark D. Rosen
, Hariharan Venkatesan
, et al.
·
ACS Medicinal Chemistry Letters
·
64
Efficient Total Syntheses of Pumiliotoxins A and B. Applications of Iodide-Promoted Iminium Ion−Alkyne Cyclizations in Alkaloid Construction
1996
·
Nan-Horng Lin
, Larry E. Overman
, et al.
·
Journal of the American Chemical Society
·
61
Enantioselective Total Syntheses of Allopumiliotoxins 267A, 323B‘, and 339A. Application of Iodide-Promoted Iminium Ion−Alkyne Cyclizations for Forming Allopumiliotoxin A Alkaloids
1996
·
Christian Caderas
, Renee Lett
, et al.
·
Journal of the American Chemical Society
·
52
Studies toward the total synthesis of (+)-ptilomycalin A. Use of a tethered Biginelli condensation for the preparation of an advanced tricyclic intermediate
1993
·
Larry E. Overman
, Michael H. Rabinowitz
·
The Journal of Organic Chemistry
·
50
Prolyl hydroxylase inhibition corrects functional iron deficiency and inflammation‐induced anaemia in rats
2015
·
Terrance D Barrett
, Heather L Palomino
, et al.
·
British Journal of Pharmacology
·
47
A One-Step Synthesis of 2,4-Unsubstituted Quinoline-3-carboxylic Acid Esters from o-Nitrobenzaldehydes
2010
·
Hariharan Venkatesan
, Frances M. Hocutt
, et al.
·
The Journal of Organic Chemistry
·
47
Discovery of the first known small-molecule inhibitors of heme-regulated eukaryotic initiation factor 2α (HRI) kinase
2009
·
Mark D. Rosen
, Craig R. Woods
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
41
Physiological Control of Nitric Oxide in Neuronal BACE1 Translation by Heme-Regulated eIF2α Kinase HRI Induces Synaptogenesis
2015
·
Gerard Ill-Raga
, Marta Tajes
, et al.
·
Antioxidants and Redox Signaling
·
36
Identification and Optimization of Anthranilic Sulfonamides as Novel, Selective Cholecystokinin-2 Receptor Antagonists
2006
·
Brett D. Allison
, Victor K. Phuong
, et al.
·
Journal of Medicinal Chemistry
·
36
Preclinical Characterization of Vadadustat (AKB-6548), an Oral Small Molecule Hypoxia-Inducible Factor Prolyl-4-Hydroxylase Inhibitor, for the Potential Treatment of Renal Anemia
2022
·
Anna Zuk
, Zhihai Si
, et al.
·
Journal of Pharmacology and Experimental Therapeutics
·
33
PDF
Substrate Specificity and Novel Selective Inhibitors of TNF-α Converting Enzyme (TACE) from Two-Dimensional Substrate Mapping
2005
·
Millard Lambert
, R. Blackburn
, et al.
·
Combinatorial Chemistry & High Throughput Screening
·
26
Biosynthetic studies of marine lipids. 39. 19-Norsterols: the course of C-19 methyl elimination
1992
·
Michael H. Rabinowitz
, Carl Djerassi
·
Journal of the American Chemical Society
·
24
A convenient synthesis of pyrazolidine and 3‐amino‐6,7‐dihydro‐1H,5H‐pyrazolo[1,2‐a] pyrazol‐1‐one
2001
·
Eric E. Boros
, Frédéric Bouvier
, et al.
·
Journal of Heterocyclic Chemistry
·
23
Glutamatergic stimulation induces GluN2B translation by the nitric oxide-Heme-Regulated eIF2α kinase in cortical neurons
2016
·
Eva Ramos-Fernández
, Marta Tajes
, et al.
·
Oncotarget
·
21
PDF
N-Hydroxyformamide peptidomimetics as TACE/Matrix metalloprotease inhibitors: oral activity via P1′ isobutyl substitution
2001
·
David L. Musso
, Marc W. Andersen
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
20
Hantzsch Synthesis of Pyrazolo[1‘,2‘:1,2]pyrazolo[3,4-b]pyridines: Partial Agonists of the Calcitonin Receptor
2005
·
Eric E. Boros
, David J. Cowan
, et al.
·
The Journal of Organic Chemistry
·
18
Solid-phase/solution-phase combinatorial synthesis of neuroimmunophilin ligands
2000
·
Michael Rabinowitz
, Pierfausto Seneci
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
17
A general method for the synthesis of benzimidazole-4-sulfonamides
2009
·
Mark D. Rosen
, Zahna M. Simon
, et al.
·
Tetrahedron Letters
·
15
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Works count:
55
Citation count:
1,486
H-index:
21
I10-index:
30
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