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Guillaume Le Baut

Observed names: BAUT, Guillaume LE, Baut, Guillaume Le, G LEBAUT, G Le Baut, G. LE BAUT, G. Le Baut, G. Y. LE BAUT, GUILLAUME LE BAUT, Guillaume Baut, Guillaume Le baut, Guillaume LeBaut, Guillaume le Baut, LE BAUT, Guillaume, Le Baut G, Le Baut, Guillaume
ORCID: 0000-0002-9442-4554
Observed ORCID: 0000-0002-9442-4554
OpenAlex ID: A5003051645
Effects of tumour necrosis factor-α synthesis inhibitors on rat trinitrobenzene sulphonic acid-induced chronic colitis
2001 · Christine Bobin-Dubigeon, Xavier Collin, et al. · European Journal of Pharmacology · 83
Synthesis and biological evaluation of 5-[(aryl)(1H-imidazol-1-yl)methyl]-1H-indoles: Potent and selective aromatase inhibitors
2005 · Marie-Pierre Lézé, Marc Le Borgne, et al. · Bioorganic & Medicinal Chemistry Letters · 71
Synthesis and antifungal activities of new fluconazole analogues with azaheterocycle moiety
2007 · Nicolas Lebouvier, Fabrice Pagniez, et al. · Bioorganic & Medicinal Chemistry Letters · 70
New anti-inflammatory N-pyridinyl(alkyl)phthalimides acting as tumour necrosis factor-α production inhibitors
2001 · Xavier Collin, Jean-Michel Robert, et al. · European Journal of Medicinal Chemistry · 69
2- and 3-[(Aryl)(azolyl)methyl]indoles as Potential Non-steroidal Aromatase Inhibitors
2004 · Marie-Pierre Lézé, Marc Le Borgne, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 67
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New selective nonsteroidal aromatase inhibitors: Synthesis and inhibitory activity of 2,3 or 5-(α-azolylbenzyl)-1H-indoles
1999 · Marc Le Borgne, Pascal Marchand, et al. · Bioorganic & Medicinal Chemistry Letters · 65
Synthesis and In Vitro Evaluation of 3‐(1‐Azolylmethyl)‐1H‐indoles and 3‐(1‐Azolyl‐1‐phenylmethyl)‐1H‐indoles as Inhibitors of P450 arom
1997 · Marc Le Borgne, Pascal Marchand, et al. · Archiv der Pharmazie · 58
Potential application of plant lipid transfer proteins for drug delivery
2001 · Christine Pato, Marc Le Borgne, et al. · Biochemical Pharmacology · 51
Efficient microwave-assisted synthesis of 1-(1H-indol-1-yl)-2-phenyl-3-(1H-1,2,4-triazol-1-yl)propan-2-ols as antifungal agents
2006 · Nicolas Lebouvier, Francis Giraud, et al. · Tetrahedron Letters · 50
Preparation and pharmacological profile of 7-(α-Azolylbenzyl)-1H-indoles and indolines as new aromatase inhibitors
2003 · Pascal Marchand, Marc Le Borgne, et al. · Bioorganic & Medicinal Chemistry Letters · 37
Pyrophtalones VII. Synthèse et activité anti-inflammatoire de (pyridinyl-4)-2 indanediones-1,3 substituées sur le noyau benzénique et/ou sur l'hétérocycle
1987 · Danielle Leblois, Sylvie Piessard, et al. · European Journal of Medicinal Chemistry · 32
Synthesis and antileishmanial activity of new imidazolidin-2-one derivatives
2003 · Jean-Michel H Robert, Caroline Sabourin, et al. · European Journal of Medicinal Chemistry · 31
Synthesis of N-Pyridinyl(methyl)-1,2-dihydro-4-hydroxy-2-oxoquinoline-3-carboxamides and analogues and their anti-inflammatory activity in mice and rats
2001 · X Collin, J M Robert, et al. · Journal of Pharmacy and Pharmacology · 26
Non-acidic anti-inflammatory compounds: activity of N-(4,6-dimethyl-2-pyridinyl) benzamides and derivatives
1990 · Sylvie Robert-Piessard, Guillaume Le Baut, et al. · European Journal of Medicinal Chemistry · 23
Synthesis, Optimization, Antifungal Activity, Selectivity, and CYP51 Binding of New 2-Aryl-3-azolyl-1-indolyl-propan-2-ols
2020 · Nicolas Lebouvier, Fabrice Pagniez, et al. · Pharmaceuticals · 21
Synthesis and structure–activity relationships of N-aryl(indol-3-yl)glyoxamides as antitumor agents
2009 · Pascal Marchand, Maud Antoine, et al. · Bioorganic & Medicinal Chemistry · 21
Inhibition of Parasite Protein Kinase C by New Antileishmanial Imidazolidin-2-one Compounds
2002 · Nidia Alvarez, Sara Robledo, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 21
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Antileishmanial activities and mechanisms of action of indole-based azoles
2006 · Fabrice Pagniez, Hiam Abdala-Valencia, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 20
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Three-dimensional model of cytochrome P450 human aromatase
2005 · Cedric Loge, Marc Le Borgne, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 18
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New N -pyridinyl(methyl)-indole-2- and 3-(Alkyl)carboxamides and Derivatives Acting as Systemic and Topical Inflammation Inhibitors
2002 · Anne Breteche, Muriel Duflos, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 18
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Non-carboxylic antiinflammatory compounds. III. N-(4,6-Dimethylpyridin-2-yl)arylcarboxamides and arylthiocarboxamides acting as brain edema inhibitors
1995 · J.M.H. Robert, S Robert-Piessard, et al. · European Journal of Medicinal Chemistry · 18
New N -(Pyridin-4-yl)-(indol-3-yl)acetamides and Propanamides as Antiallergic Agents
1999 · Cecilia Menciu, Muriel Duflos, et al. · Journal of Medicinal Chemistry · 17
Non-acidic antiinflammatory compounds II. Synthesis and activity of 6-amino-2,4-lutidine derivatives
1994 · J ROBERT, S ROBERTPIESSARD, et al. · European Journal of Medicinal Chemistry · 16
Synthesis of new bifunctional chelating agents: (1R*,2R*,4S*)-4-isothiocyanatocyclohexane-1,2-diamine-N,N,N′,N′-tetrakismethanephosphonic acid (4-ICMP) and (1R*,2R*,4S*)-4-isothiocyanatocyclohexane-1,2-diamine-N,N,N′,N′-tetrakisethanephosphonic acid (4-ICEP)
1998 · Anthony Loussouarn, Muriel Duflos, et al. · Journal of the Chemical Society Perkin Transactions 1 · 15
New Route to Styrylchromones via [1-(2-Hydroxybenzoyl)alkylidene]triphenylphosphoranes
1992 · F. Zammattio, J. D. Brion, et al. · Synthesis · 14
Works count: 154
Citation count: 1,217
H-index: 18
I10-index: 38
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