Author

Grazyna Kurylko

Observed name: Kurylko, G.

Observed institution: F. Hoffmann-La Roche AG

OpenAlex ID: A5021551901

A Novel Selective Melanocortin-4 Receptor Agonist Reduces Food Intake in Rats and Mice without Producing Aversive Consequences

2000 · Stephen C. Benoit, Michael W. Schwartz, et al. · Journal of Neuroscience · 178

Opportunities and Challenges of Developing Peptide Drugs in the Pharmaceutical Industry

2009 · Waleed Danho, Joseph Swistok, et al. · Advances in experimental medicine and biology · 39

Effects of LTB4 receptor antagonism on pulmonary inflammation in rodents and non-human primates

2010 · Alexandra Hicks, Robert Goodnow, et al. · Prostaglandins & Other Lipid Mediators · 29

Structure–Activity relationship of linear peptide Bu-His-DPhe-Arg-Trp-Gly-NH2 at the human melanocortin-1 and -4 receptors: arginine substitution

2002 · Adrian Wai-Hing Cheung, Waleed Danho, et al. · Bioorganic & Medicinal Chemistry Letters · 29

Structure–Activity relationship of linear peptide Bu-His-DPhe-Arg-Trp-Gly-NH2 at the human melanocortin-1 and -4 receptors: histidine substitution

2003 · Adrian Wai-Hing Cheung, Waleed Danho, et al. · Bioorganic & Medicinal Chemistry Letters · 26

Discovery of 1-amino-4-phenylcyclohexane-1-carboxylic acid and its influence on agonist selectivity between human melanocortin-4 and -1 receptors in linear pentapeptides

2005 · Xin-Jie Chu, David Bartkovitz, et al. · Bioorganic & Medicinal Chemistry Letters · 16

Structure–Activity relationship of linear peptide Bu-His6-DPhe7-Arg8-Trp9-Gly10-NH2 at the human melanocortin-1 and -4 receptors: DPhe7 and Trp9 substitution

2003 · Waleed Danho, Joseph Swistok, et al. · Bioorganic & Medicinal Chemistry Letters · 15

Structure–activity relationship of cyclic peptide penta-c[Asp-His6-DPhe7-Arg8-Trp9-Lys]-NH2 at the human melanocortin-1 and -4 receptors: His6 substitution

2003 · Adrian Wai-Hing Cheung, Waleed Danho, et al. · Bioorganic & Medicinal Chemistry Letters · 14

Discovery of Novel and Potent Leukotriene B4Receptor Antagonists. Part 1

2010 · Robert A. Goodnow, Alexandra Hicks, et al. · Journal of Medicinal Chemistry · 10

Preparation of human Melanocortin-4 receptor agonist libraries: Linear peptides X-Y-DPhe7-Arg8-Trp(or 2-Nal)9-Z-NH2

2005 · Adrian Wai-Hing Cheung, Lida Qi, et al. · Bioorganic & Medicinal Chemistry Letters · 8

Highly Selective Cyclic Peptides for Human Melanocortin-4 Receptor (MC-4 R): Design, Synthesis, Bioactive Conformation, and Pharmacological Evaluation as an Anti-Obesity Agent

2001 · Waleed Danho, Joseph Swistok, et al. · Springer eBooks · 4

CCDC 283241: Experimental Crystal Structure Determination

2006 · Chu, Xin-Jie, Bartkovitz, D., et al. · The Cambridge Structural Database

Works count: 12

Citation count: 368

H-index: 9

I10-index: 9