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Sandeep R. Ghorpade

Observed names: GHORPADE, SANDEEP, Ghorpade, Sandeep R., Sandeep G. Ghorpade, Sandeep Ghorpade, Sandeep R Ghorpade
ORCID: 0000-0002-9311-1572
Observed ORCID: 0000-0002-9311-1572
OpenAlex ID: A5028450220
Enantioselective Synthesis of α,β-Disubstituted-β-amino Acids
2003 · Mukund P. Sibi, Prabagaran Narayanasamy, et al. · Journal of the American Chemical Society · 122
4-Aminoquinolone Piperidine Amides: Noncovalent Inhibitors of DprE1 with Long Residence Time and Potent Antimycobacterial Activity
2014 · Maruti Naik, Vaishali Humnabadkar, et al. · Journal of Medicinal Chemistry · 96
Recent developments of imidazo[1,2- a ]pyridine analogues as antituberculosis agents
2023 · Sauvik Samanta, Sumit Kumar, et al. · RSC Medicinal Chemistry · 79
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Thiazolopyridine Ureas as Novel Antitubercular Agents Acting through Inhibition of DNA Gyrase B
2013 · Manoj G. Kale, Anandkumar Raichurkar, et al. · Journal of Medicinal Chemistry · 67
A Convenient Method for the Conversion of N-Acyloxazolidinones to Hydroxamic Acids
2002 · Mukund P. Sibi, Hikaru Hasegawa, et al. · Organic Letters · 55
Thiazolopyridone ureas as DNA gyrase B inhibitors: Optimization of antitubercular activity and efficacy
2013 · Ramesh R. Kale, Manoj G. Kale, et al. · Bioorganic & Medicinal Chemistry Letters · 43
Spiropyrimidinetrione DNA Gyrase Inhibitors with Potent and Selective Antituberculosis Activity
2022 · Preshendren Govender, Rudolf Müller, et al. · Journal of Medicinal Chemistry · 36
Whole cell screen based identification of spiropiperidines with potent antitubercular properties
2015 · Subramanyam J. Tantry, Giulia Degiacomi, et al. · Bioorganic & Medicinal Chemistry Letters · 33
2-Phenylindole and Arylsulphonamide: Novel Scaffolds Bactericidal against Mycobacterium tuberculosis
2014 · Maruti Naik, Sandeep Ghorpade, et al. · ACS Medicinal Chemistry Letters · 29
1,3-Diarylpyrazolyl-acylsulfonamides as Potent Anti-tuberculosis Agents Targeting Cell Wall Biosynthesis in Mycobacterium tuberculosis
2021 · Lutete Peguy Khonde, Rudolf Müller, et al. · Journal of Medicinal Chemistry · 26
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Spiropyrimidinetriones: a Class of DNA Gyrase Inhibitors with Activity against Mycobacterium tuberculosis and without Cross-Resistance to Fluoroquinolones
2022 · Gregory S. Basarab, Sandeep Ghorpade, et al. · Antimicrobial Agents and Chemotherapy · 24
Enzymatic kinetic resolution studies of racemic 4-hydroxycyclopent-2-en-1-one using Lipozyme IM®
1999 · Sandeep R Ghorpade, Kulbhushan B Bastawade, et al. · Tetrahedron Asymmetry · 24
Novel Antitubercular 6-Dialkylaminopyrimidine Carboxamides from Phenotypic Whole-Cell High Throughput Screening of a SoftFocus Library: Structure–Activity Relationship and Target Identification Studies
2017 · Colin R. Wilson, Richard K. Gessner, et al. · Journal of Medicinal Chemistry · 23
2,8-Disubstituted-1,5-naphthyridines as Dual Inhibitors of Plasmodium falciparum Phosphatidylinositol-4-kinase and Hemozoin Formation with In Vivo Efficacy
2024 · Godwin Akpeko Dziwornu, Donald Seanego, et al. · Journal of Medicinal Chemistry · 22
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Antitubercular 2-Pyrazolylpyrimidinones: Structure–Activity Relationship and Mode-of-Action Studies
2021 · Candice Soares de Melo, Vinayak Singh, et al. · Journal of Medicinal Chemistry · 21
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Desymmetrization of meso-cyclopenten-cis-1,4-diol to 4-(R)-hydroxycyclopent-2-en-1-(S)-acetate by irreversible transesterification using Chirazyme®
1999 · Sandeep R Ghorpade, Rajendra K Kharul, et al. · Tetrahedron Asymmetry · 16
Binding of Matrix Metalloproteinase Inhibitors to Extracellular Matrix: 3D‐QSAR Analysis
2008 · Yufen Zhang, Viera Lukacova, et al. · Chemical Biology & Drug Design · 11
Simple, Efficient Chemoenzymatic Synthesis of (S)-5-(tert-Butyldimethylsilyloxy)-2-cyclohexenone and Enantiomeric Ketone Intermediates of 19-Nor-1α,25-dihydroxyvitamin D3
2001 · Uttam R. Kalkote, Sandeep R. Ghorpade, et al. · The Journal of Organic Chemistry · 11
A Convenient Synthesis of 5-substituted 2-amino-1,3,4-oxadiazoles from Corresponding Acylthiosemicarbazides Using iodine and Oxone®
2013 · Vikas N. Shinde, Bheemarao G. Ugarkar, et al. · Journal of Chemical Research · 10
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A practical and scalable process for 4-(R)-hydroxycyclopent-2-en-1-(S)-acetate by desymmetrization of meso-cyclopent-2-en-1,4-diacetate catalyzed by Trichosporon beigelii (NCIM 3326), a cheap biocatalyst
2000 · Uttam R Kalkote, Sandeep R Ghorpade, et al. · Tetrahedron Asymmetry · 10
Efficient Synthesis of Optically Pure (4R,6S)-4-(tert-Butyldimethylsilyloxy)- 6-(hydroxymethyl)tetrahydropyran-2-one and Its Enantiomer
2001 · Sandeep R. Ghorpade, Uttam R. Kalkote, et al. · The Journal of Organic Chemistry · 7
Novel Inhibitors of Plasmodium Phosphatidylinositol 4-kinase IIIβ with Low Propensity for Resistance: Life Cycle Stage Activity and In Vivo Efficacy in a Humanized Mouse Malaria Infection Model
2025 · Godwin A. Dziwornu, Mmakwena M. Mmonwa, et al. · Journal of Medicinal Chemistry · 5
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1,3-Diarylpyrazolyl-acylsulfonamides Target HadAB/BC Complex in Mycobacterium tuberculosis
2022 · Vinayak Singh, Anna E. Grzegorzewicz, et al. · ACS Infectious Diseases · 5
Structure−Activity relationship and optimization of drug-like properties of antituberculosis 3-(4,4-dimethyl-1,4-azasilinane)methylpyrazole MmpL3 inhibitors
2026 · Lutete Peguy Khonde, Nashied Peton, et al. · European Journal of Medicinal Chemistry · 1
Optimization of 2,8-Diaryl-1,5-naphthyridines as Plasmodium falciparum Phosphatidylinositol 4-Kinase Inhibitors with Improved ADME Profiles and In Vivo Efficacy
2025 · Godwin A. Dziwornu, Donald Seanego, et al. · Journal of Medicinal Chemistry · 1
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Works count: 33
Citation count: 777
H-index: 16
I10-index: 20
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